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Monophthalates of betulinic acid and related pentacyclic triterpenes inhibit efficiently the SOS-mediated nucleotide exchange and impact PI3K/AKT signaling in oncogenic K-RAS4B proteins. Gerrit E. Benary, Frank Kilgenstein, Sascha Koller, Jürgen Scherkenbeck*. ChemRxiv 2024, DOI 10.26434/chemrxiv-2024-x4tfq. RSC Adv. 2025, 15, 883-895.
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Enabling antibiotic research: towards selective peptide deformylase inhibitors. Nathalie Bachmann, André Schultz, Manuela Zouatom, Tianyi Zhou, Carsten Degenhart, Uwe Koch, Sina Schäkermann, Julia Hüning, Sascha Heinrich, Michael Dal Molin, Mia-Lisa Zischinsky, Sylvain Tourel, Anne-Kathrin Kleb, Jan Rybniker, Bert M. Klebl, Jürgen Scherkenbeck, Julia E. Bandow1. Doi: https://doi.org/10.1101/2025.09.18.677056
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A highly efficient access to new antibacterial actinonin derivatives via Ugi four-component reaction. Manuela Zouatom, Tianji Zhou, André Schultz, Nathalie Bachmann, Carsten Degenhart, Michael Dal Molin, Uwe Koch, Jan Rybniker, Bert Klebl, Julia Elisabeth Bandow, Jürgen Scherkenbeck. Doi: 10.26434/chemrxiv-2025-kf42k